Lysine-targeted covalent inhibitor design
Mutant-selective AKT inhibition via lysine targeting and neo-zinc chelation.
Nature. 2025.
Craven GB, Chu H, Sun JD, Carelli JD, Coyne B, Chen H, Chen Y, Ma X, Das S, Kong W, Zajdlik AD, Yang KS, Reisberg SH, Thompson PA, Lipford JR, Taunton J.